发明名称 |
CRYSTALLINE SOLVATES AND COMPLEXES OF (IS) -1, 5-ANHYDRO-L-C- (3- ( (PHENYL) METHYL) PHENYL) -D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES |
摘要 |
The present invention relates to physical crystal structures of a compound of the formula I:
wherein R 1 , R 2 , R 2a , R 3 and R 4 are as defined herein, especially
pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures. |
申请公布号 |
HRP20141007(T1) |
申请公布日期 |
2014.12.05 |
申请号 |
HR2014P001007T |
申请日期 |
2014.10.21 |
申请人 |
ASTRAZENECA AB |
发明人 |
GOUGOUTAS, JACK Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT P.;BIEN, JEFFREY T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN ANTHONY;NIRSCHL, ALEXANDRA A.;SINGH, JANAK;DIMARCO, JOHN D. |
分类号 |
C07H7/04;A61K31/70;A61P3/10 |
主分类号 |
C07H7/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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