发明名称 CRYSTALLINE SOLVATES AND COMPLEXES OF (IS) -1, 5-ANHYDRO-L-C- (3- ( (PHENYL) METHYL) PHENYL) -D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 The present invention relates to physical crystal structures of a compound of the formula I: wherein R 1 , R 2 , R 2a , R 3 and R 4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
申请公布号 HRP20141007(T1) 申请公布日期 2014.12.05
申请号 HR2014P001007T 申请日期 2014.10.21
申请人 ASTRAZENECA AB 发明人 GOUGOUTAS, JACK Z.;LOBINGER, HILDEGARD;RAMAKRISHNAN, SRIVIDYA;DESHPANDE, PRASHANT P.;BIEN, JEFFREY T.;LAI, CHIAJEN;WANG, CHENCHI;RIEBEL, PETER;GROSSO, JOHN ANTHONY;NIRSCHL, ALEXANDRA A.;SINGH, JANAK;DIMARCO, JOHN D.
分类号 C07H7/04;A61K31/70;A61P3/10 主分类号 C07H7/04
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