发明名称 CRYSTALLINE FORM OF N,N-DICYCLOPROPYL-4-(1,5-DIMETHYL-1 H-PYRAZOL-3-YLAMINO)-6-ETHYL-1 -METHYL-1,6-DIHYRDROIMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDINE-7-CARBOXAMIDE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISORDERS
摘要 Crystalline form, Form N-2, of N, Ndicyclopropyl-4-(l,5-dimethyl-1 Hpyrazol-3-ylamino)-6-ethyl-l-methyl-l,6-dihydroimidazo[4,5- d]pyrrolo[2,3-b]pyridine-7-carboxamide (Compound I) is provided. Also provided are a pharmaceutical composition and an oral dosage form comprising Form N-2 of Compound I as well as a method of using the Form N-2 of Compound I in the treatment of myeloproliferative disorders, which include polycythaemia vera, thrombocythaemia and primary myelofibrosis.
申请公布号 WO2014193881(A1) 申请公布日期 2014.12.04
申请号 WO2014US39657 申请日期 2014.05.28
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 TAMEZE, SHELLA
分类号 C07D471/14;A61K31/437;A61P35/00;A61P37/00 主分类号 C07D471/14
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