发明名称 |
PROCESS FOR MAKING CGRP RECEPTOR ANTAGONISTS |
摘要 |
<p>The invention encompasses a novel process for making piperidinone carboxamide indane and azainane derivatives, which are CGRP receptor antagonists useful for the treatment of migraine, utilizing a highly effective spiroacid synthesis.</p> |
申请公布号 |
KR20140138705(A) |
申请公布日期 |
2014.12.04 |
申请号 |
KR20147025146 |
申请日期 |
2013.03.13 |
申请人 |
MERCK SHARP & DOHME CORP. |
发明人 |
BELYK KEVIN M.;CLEATOR EDWARD;KUO SHEN CHUN;MALIGRES PETER EMMANUEL;XIANG BANGPING;YASUDA NOBUYOSHI;YIN JIANGUO |
分类号 |
C07D401/14;A61K31/519;C07D401/12 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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