发明名称 |
ANHYDROUS POLYMORPHS OF (2R,3S,4R,5R)-5-(6-(CYCLOPENTYLAMINO)-9H-PURIN-9-YL)-3,4-DIHYDROXYTETRAHYDROFURAN-2-YL) } METHYL NITRATE AND PROCESSES OF PREPARATION THEREOF |
摘要 |
<p>The present invention provides novel anhydrous polymorph forms of 2R,3S,4R,5R)-5-(6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl nitrate (Compound A). The present invention also provides processes for preparation of the anhydrous polymorphic forms of compound A.</p> |
申请公布号 |
EP2807178(A1) |
申请公布日期 |
2014.12.03 |
申请号 |
EP20130741502 |
申请日期 |
2013.01.25 |
申请人 |
INOTEK PHARMACEUTICALS CORPORATION |
发明人 |
MCVICAR, WILLIAM, K. |
分类号 |
C07H19/167;A61K31/7076;A61P27/02;A61P27/06 |
主分类号 |
C07H19/167 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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