发明名称 |
CRYSTALLINE FORMS AND TWO SOLVATED FORMS OF 4-AMINO-5-FLUORO-3-[5-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE LACTIC ACID SALTS |
摘要 |
<p>Crystalline forms or polymorphs of 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one lactic acid salts, as well as to methods of making the same, pharmaceutical compositions comprising the same and methods of treatment using the same.</p> |
申请公布号 |
EP2257544(B1) |
申请公布日期 |
2014.12.03 |
申请号 |
EP20090721534 |
申请日期 |
2009.03.18 |
申请人 |
NOVARTIS AG |
发明人 |
GIRON, DANIELLE;HAMMERSCHMIDT, WALTER;PIECHON, PHILIPPE;POLASEK, JOHANNE;SCHREINER, ANDREAS;STOWASSER, FRANK |
分类号 |
C07D401/14;A61K31/496;A61P35/00 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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