发明名称 |
SUBSITUTED ALIPHANES, CYCLOPHANES, HETERAPHANES, HETEROPHANES, HETERO-HETERAPHANES AND METALLOCENES USEFUL FOR TREATING HCV INFECTIONS |
摘要 |
Provided is a compound having a structure selected from the group consisting of:
which are intermediates in the preparation of Carbamic acid,
N,N'-[tricyclo[8.2.2.24,7]hexadeca-4,6,10,12,13,15-hexaene-5,11-diyl bis [1H-benzimidazole-6,2-diyl[(2S,3aS,7aS)-octahydro-1H-indole-2,1-diyl][(1S)-1-(1-methylethyl)-2-oxo-2,1-ethane diyl]]] bis-, C,C'-dimethyl ester, which is a Hepatitis C virus NS5a (HCV NS5a) protease replication inhibitor |
申请公布号 |
EP2714036(A4) |
申请公布日期 |
2014.11.12 |
申请号 |
EP20120793566 |
申请日期 |
2012.05.29 |
申请人 |
ACHILLION PHARMACEUTICALS, INC. |
发明人 |
WILES, JASON ALLAN;WANG, QIUPING;HASHIMOTO, AKIHIRO;PAIS, GODWIN;CHEN, DAWEI;WANG, XIANGZHU;GADHACHANDA, VENKAT;PHADKE, AVINASH;DESHPANDE, MILIND |
分类号 |
C07F17/02;A61K31/4164;A61K31/4178;A61P31/00;A61P31/12;C07D401/14;C07D403/14;C07D413/14;C07D417/14;C07D471/08;C07D471/14;C07D491/10;C07D519/00 |
主分类号 |
C07F17/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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