发明名称 |
COMPOUNDS, THEIR PHARMACEUTICAL COMPOSITIONS AND THEIR USES AS IDH1 MUTANTS INHIBITORS FOR TREATING CANCERS |
摘要 |
Provided are compounds of formula (I), wherein X, Y, Z, W, V, R2, R3 and m are defined as in the description. Their pharmaceutical compositions and their uses for treating cancers are also provided. |
申请公布号 |
EP2721033(A4) |
申请公布日期 |
2014.11.05 |
申请号 |
EP20120799802 |
申请日期 |
2012.06.18 |
申请人 |
AGIOS PHARMACEUTICALS, INC. |
发明人 |
CAO, SHELDON;POPOVICI-MULLER, JANETA;SALITURO, FRANCESCO G.;SAUNDERS, JEFFREY O.;TAN, XUEFEI;TRAVINS, JEREMY;YAN, SHUNQI;YE, ZHIXIONG |
分类号 |
C07D491/052;A61K31/496;A61P35/00;C07D217/26;C07D413/04;C07D519/00 |
主分类号 |
C07D491/052 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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