发明名称 NEW CRYSTALLINE FORMS OF APIXABAN AND A METHOD OF THEIR PREPARATION
摘要 The present invention relates to new crystalline forms of apixaban of formula (I), chemically 1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H- pyrazolo[3,4-c]pyridine-3-carboxamide of formula I, and a method of their preparation. The concerned forms are AP3, AP4 and AP5.
申请公布号 WO2014173377(A2) 申请公布日期 2014.10.30
申请号 WO2014CZ00041 申请日期 2014.04.23
申请人 ZENTIVA, K.S. 发明人 KISS, VIOLETTA;DAMMER, ONDREJ;KREJCIK, LUKAS;HEJTMANKOVA, LUDMILA
分类号 C07D471/04;A61K31/437 主分类号 C07D471/04
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