发明名称 |
CRYSTALLINE FORM OF CABAZITAXEL AND PROCESS FOR PREPARING THE SAME |
摘要 |
The present invention relates to a novel crystalline ethyl acetate solvate form of cabazitaxel or 4α-acetoxy-2α-benzoyloxy-5&bgr;,20-epoxy-1&bgr;-hydroxy-7&bgr;,10&bgr;-dimethoxy-9-oxo-11-taxen-13α-yl(2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate and process for preparing the same. |
申请公布号 |
EP2791122(A1) |
申请公布日期 |
2014.10.22 |
申请号 |
EP20120815825 |
申请日期 |
2012.12.11 |
申请人 |
AVENTIS PHARMA S.A. |
发明人 |
DIDIER, ERIC;TREMAUDEUX, NICOLAS;ZASKE, LIONEL |
分类号 |
C07D305/14;A61K31/337;A61P35/00 |
主分类号 |
C07D305/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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