发明名称 Sustained release compositions containing progesterone receptor modulators
摘要 Disclosed are sustained release compositions for vaginal or transdermal administration that contain a progesterone receptor modulator such as CDB-2914 (also referred to as VA-2914), and methods of using them for long term contraception or therapeutic purposes. Also disclosed are methods for making the compositions.
申请公布号 US8865200(B2) 申请公布日期 2014.10.21
申请号 US200511631877 申请日期 2005.07.08
申请人 Laboratoire HRA Pharma 发明人 Sitruk-Ware Regine;Tsong Yun-Yen
分类号 A61F6/06;A61K31/56;A61K47/30;A61K47/24;A61K9/00;A61F6/08 主分类号 A61F6/06
代理机构 Lerner, David, Littenberg, Krumholz & Mentlik, LLP 代理人 Lerner, David, Littenberg, Krumholz & Mentlik, LLP
主权项 1. A vaginal ring composition comprising a synthetic polymer having contained therein a contraceptively effective amount of a steroid comprising a progesterone receptor modulator (PRM), with the proviso that the progesterone receptor modulator is not an androgen, selected androgen receptor modulator, estrogen, or selected estrogen receptor modulator.
地址 FR