发明名称 |
DIAZACARBAZOLES AND METHODS OF USE |
摘要 |
<p>PROBLEM TO BE SOLVED: To provide compounds which are useful as kinase inhibitors, more specifically useful as checkpoint kinase 1 (chk1), thus useful as cancer therapeutics.SOLUTION: The invention relates to 1,5-diazacarbazole compounds of the following formula.</p> |
申请公布号 |
JP2014196309(A) |
申请公布日期 |
2014.10.16 |
申请号 |
JP20140103195 |
申请日期 |
2014.05.19 |
申请人 |
GENENTECH INC |
发明人 |
HAZEL JOAN DYKE;EMANUELA GANCIA;GAZZARD LEWIS J;SIMON CHARLS GOODACRE;LYSSIKATOS JOSEPH P;CALUM MACLEOD;KAREN WILLIAMS;CHEN HUIFEN |
分类号 |
C07D471/14;A61K31/496;A61K31/519;A61K45/00;A61P35/00;A61P35/02 |
主分类号 |
C07D471/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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