摘要 |
<p>THE PRESENT INVENTION RELATES TO 1-ARYL-3-ANILINE-5-ALKYL-1,2,4-TRIAZOLE DERIVATIVES AND ANALOGUES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PROCESSES FOR PREPARING THEM, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY, ACCORDING TO FORMULA (I). THE INVENTION PARTICULARLY RELATES TO POTENT POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS, SUCH POSITIVE ALLOSTERIC MODULATOR HAVING THE CAPABILITY TO INCREASE THE EFFICACY OF NICOTINIC RECEPTOR AGONISTS. (NO SUITABLE</p> |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
MACDONALD, GREGOR, JAMES;THURING, JOHANNES, WILHELMUS, JOHN F.;STANISLAWSKI, PAULINE, CAROL;ZHUANG, WEI;VAN ROOSBROECK, YVES, EMIEL, MARIA;VAN DEN KEYBUS, FRANS, ALFONS, MARIA |