| 发明名称 |
CYCLIC UREA DERIVATIVES AS ANDROGEN RECEPTOR ANTAGONISTS |
| 摘要 |
<p>The present invention is directed to compounds of formula (I) wherein R1, R2, R3, and A are defined herein. The present invention also provides for pharmaceutical compositions comprising a compound of formula (I) as well as to the use of such compounds as androgen receptor antagonists for the treatment of diseases and conditions mediated by the androgen receptor, such as prostate cancer.</p> |
| 申请公布号 |
EP2788330(A1) |
申请公布日期 |
2014.10.15 |
| 申请号 |
EP20120813983 |
申请日期 |
2012.12.03 |
| 申请人 |
NOVARTIS AG |
发明人 |
BOCK, MARK;CHIKKANNA, DINESH;GERSPACHER, MARC;KHAIRNAR, VINAYAK;LAGU, BHARAT;PANDIT, CHETAN |
| 分类号 |
C07D235/02;A61K31/4184;A61K31/4188;A61P5/26;A61P35/00;C07D235/26;C07D401/04;C07D401/12;C07D401/14;C07D405/04;C07D405/12;C07D409/04;C07D491/052 |
主分类号 |
C07D235/02 |
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