发明名称 |
PIPERAZINYL PYRIMIDINE DERIVATIVES, PREPARATION METHOD AND USE THEREOF |
摘要 |
Provided are piperazinyl pyrimidine derivatives of formula I having CCR 4 antagonism, and the preparation method, pharmaceutical composition and use thereof in the preparation of a medicament. The medicament is useful for the treatment and prevention of CCR 4 -related diseases. |
申请公布号 |
KR20140121441(A) |
申请公布日期 |
2014.10.15 |
申请号 |
KR20147022723 |
申请日期 |
2013.01.15 |
申请人 |
INSTITUTE OF PHARMACOLOGY AND TOXICOLOGY ACADEMY OF MILITARY MEDICAL SCIENCES P.L.A. CHINA;PEKING UNIVERSITY |
发明人 |
LI SONG;WANG YING;XIAO JUNHAI;MA DALONG;GONG HONGWEI;QI HUI;WANG LILI;LING XIAOMEI;ZHENG ZHIBING;ZHANG YANG;ZHONG WU;LI MEINA;XIE YUNDE;XU ENQUAN;LI XINGZHOU;MA JING;ZHAO GUOMING;ZHOU XINBO;WANG XIAOKUI;LIU HONGYING |
分类号 |
C07D403/04;A61K31/506;A61P11/06;A61P17/00;C07D403/14 |
主分类号 |
C07D403/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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