发明名称 PIPERAZINYL PYRIMIDINE DERIVATIVES, PREPARATION METHOD AND USE THEREOF
摘要 Provided are piperazinyl pyrimidine derivatives of formula I having CCR 4 antagonism, and the preparation method, pharmaceutical composition and use thereof in the preparation of a medicament. The medicament is useful for the treatment and prevention of CCR 4 -related diseases.
申请公布号 KR20140121441(A) 申请公布日期 2014.10.15
申请号 KR20147022723 申请日期 2013.01.15
申请人 INSTITUTE OF PHARMACOLOGY AND TOXICOLOGY ACADEMY OF MILITARY MEDICAL SCIENCES P.L.A. CHINA;PEKING UNIVERSITY 发明人 LI SONG;WANG YING;XIAO JUNHAI;MA DALONG;GONG HONGWEI;QI HUI;WANG LILI;LING XIAOMEI;ZHENG ZHIBING;ZHANG YANG;ZHONG WU;LI MEINA;XIE YUNDE;XU ENQUAN;LI XINGZHOU;MA JING;ZHAO GUOMING;ZHOU XINBO;WANG XIAOKUI;LIU HONGYING
分类号 C07D403/04;A61K31/506;A61P11/06;A61P17/00;C07D403/14 主分类号 C07D403/04
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