主权项 |
1. A compound of Formula (1):wherein
each of X1 and X2 independently, is halo or OSO2Ra, in which Ra is alkyl, alkenyl, or alkynyl; Q is cycloalkyl, cycloalkenyl, heterocycloalkenyl, aryl, or heteroaryl, each of which, independently, is optionally substituted with alkyl, alkenyl, alkynyl, cycloalkyl, heterocycloalkyl, cycloalkenyl, heterocycloalkenyl, aryl, heteroaryl, halo, nitro, oxo, —CH═NH, cyano, alkyl-Rb, CH═NORb, ORb, OC(O)Rb, OC(O)ORb, OC(O)SRb, SRb, C(O)Rb, C(O)ORb, C(O)SRb, C(O)NRcRd, SORb, SO2Rb, NRcRd, alkyl-NRcRd, or N(ROC(O)Rd, in which each of Rb, Rc, and Rd, independently, is H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocycloalkyl, aryl, heteroaryl, halo, cyano, nitro, amino, hydroxyl, alkylamino, haloalkyl, or alkoxy; Z is deleted or (CH2)m in which m is an integer from 1 to 10; and each of R1 and R2 independently, is H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocycloalkyl, cycloalkenyl, heterocycloalkenyl, aryl, heteroaryl, halo, nitro, oxo, —CH═NH, cyano, alkyl-Rb, CH═NORb, ORb, OC(O)Rb, OC(O)ORb, OC(O)SRb, SRb, C(O)Rb, C(O)ORb, C(O)SRb, C(O)NRcRd, SORb, SO2Rb, NRcRd, alkyl-NRcRd, or N(Rc)C(O)Rd. |