发明名称 6-(5-HYDROXY-1H-PYRAZOL-1-YL)NICOTINAMIDE DERIVATIVES AND THEIR USE AS PHD INHIBITORS
摘要 The present invention provides compounds of formula (I) which are useful as inhibitors of PHD, pharmaceutical compositions thereof, methods for treatment of conditions associated with HIF, processes for making the compounds and intermediates thereof.
申请公布号 WO2014160810(A1) 申请公布日期 2014.10.02
申请号 WO2014US31918 申请日期 2014.03.26
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;BROWN, JASON, W.;DAVIS, MELINDA;IVETAC, ANTHONY;JONES, BENJAMIN;KIRYANOV, ANDRE, A.;KUEHLER, JON;LANIER, MARION;MIURA, JOANNE;MURPHY, SEAN;WANG, XIAOLUN 发明人 BROWN, JASON, W.;DAVIS, MELINDA;IVETAC, ANTHONY;JONES, BENJAMIN;KIRYANOV, ANDRE, A.;KUEHLER, JON;LANIER, MARION;MIURA, JOANNE;MURPHY, SEAN;WANG, XIAOLUN
分类号 C07D401/14;A61K31/443;A61K31/4433;A61K31/4436;A61K31/4439;A61K31/4545;A61K31/496;C07D401/04;C07D405/14;C07D413/14;C07D417/14;C07D471/08;C07D487/06;C07D487/10;C07D491/10 主分类号 C07D401/14
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