发明名称 PROCESS FOR THE MANUFACTURE OF (R)-5-[2-(5,6-DIETHYLINDAN-2-YLAMINO)-1-HYDROXYETHYL]-8-HYDROXY-(1H)-QUINOLIN-2-ONE
摘要 The present invention provides an efficient process for manufacturing (R)-5-[2-(5,6-diethyl-indan-2-yl-amino)-1-hydroxyethyl]-8-hydroxy-(1H)-quinolin-2-one, commonly known as indacaterol, or a pharmaceutically acceptable salt thereof, comprising intermediates of synthesis of Formula (II) and Formula (III).
申请公布号 WO2014154841(A1) 申请公布日期 2014.10.02
申请号 WO2014EP56229 申请日期 2014.03.27
申请人 LABORATORIOS LESVI, S.L. 发明人 DALMASES BARJOAN, PERE;HUGUET CLOTET, JUAN;CAPDEVILLA, ENRIC
分类号 C07D215/26 主分类号 C07D215/26
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