发明名称 ACYCLIC CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS
摘要 The instant invention provides compounds of formula I which are JAK inhibitors, and as such are useful for the treatment of JAK-mediated diseases such as rheumatoid arthritis, asthma, COPD and cancer.
申请公布号 WO2014146493(A1) 申请公布日期 2014.09.25
申请号 WO2014CN00299 申请日期 2014.03.19
申请人 MERCK SHARP & DOHME CORP.;DINSMORE, CHRISTOPHER;FULLER, PETER;GUERIN, DAVID;KATZ, JASON DAVID;THOMPSON, CHRISTOPHER F.;FALCONE, DANIELLE;DENG, WEI;TORRES, LUIS;ZENG, HONGBO;BAI, YUNFENG;FU, JIANMIN;KONG, NORMAN;LIU, YUMEI;ZHENG, ZHIXIANG 发明人 DINSMORE, CHRISTOPHER;FULLER, PETER;GUERIN, DAVID;KATZ, JASON DAVID;THOMPSON, CHRISTOPHER F.;FALCONE, DANIELLE;DENG, WEI;TORRES, LUIS;ZENG, HONGBO;BAI, YUNFENG;FU, JIANMIN;KONG, NORMAN;LIU, YUMEI;ZHENG, ZHIXIANG
分类号 C07D487/04;A61K31/437;A61K31/4375;A61P25/00;A61P35/00;A61P37/00;C07D487/08;C07D487/14 主分类号 C07D487/04
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