发明名称 CYCLOALKYL NITRILE PYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS
摘要 The instant invention provides compounds of formula I which are JAK inhibitors, and as such are useful for the treatment of JAK-mediated diseases such as rheumatoid arthritis, asthma, COPD and cancer.
申请公布号 WO2014146246(A1) 申请公布日期 2014.09.25
申请号 WO2013CN72867 申请日期 2013.03.19
申请人 MERCK SHARP & DOHME CORP.;CHILDERS, MATTHEW L.;DINSMORE, CHRISTOPHER;FULLER, PETER H.;GUERIN, DAVID J.;KATZ, JASON DAVID;PU, QINGLIN;SCOTT, MARK E.;THOMPSON, CHRISTOPHER F.;ZHANG, HONGJUN;CAI, JIAQIANG;DU, XIAOXING;WANG, CHONGGANG;KONG, NORMAN;LIU, YUMEI 发明人 CHILDERS, MATTHEW L.;DINSMORE, CHRISTOPHER;FULLER, PETER H.;GUERIN, DAVID J.;KATZ, JASON DAVID;PU, QINGLIN;SCOTT, MARK E.;THOMPSON, CHRISTOPHER F.;ZHANG, HONGJUN;CAI, JIAQIANG;DU, XIAOXING;WANG, CHONGGANG;KONG, NORMAN;LIU, YUMEI
分类号 C07D401/14;A61K31/495;A61P29/00;C07D471/04 主分类号 C07D401/14
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