发明名称 HCV NS3 PROTEASE INHIBITORS
摘要 The present invention relates to macrocyclic compounds of formula (I) that are useful as inhibitors of the hepatitis C virus (HCV) NS3 protease, their synthesis, and their use for treating or preventing HCV infections.
申请公布号 EP2780026(A2) 申请公布日期 2014.09.24
申请号 EP20120850713 申请日期 2012.11.09
申请人 MERCK SHARP & DOHME CORP.;MERCK CANADA INC.;ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.R.L. 发明人 RUDD, MICHAEL, T.;MCCAULEY, JOHN;LIVERTON, NIGEL;GRISE-BARD, CHRISTIANE;BROUCHU, MARIE-CHRISTINE;CHARRON, SYLVIE;AULAKH, VIRENDER;BACHAND, BENOIT;BEAULIEU, PATRICK;ZAGHDANE, HELMI;HAN, YONGXIN;FERRARA, MARCO;HARPER, STEVEN;SUMMA, VINCENZO;CHACKALAMANNIL, SAMUEL;VENKATRAMAN, SRIKANTH;SHAH, UNMESH;VELAZQUEZ, FRANCISCO
分类号 A61K38/12;A61P31/12;A61P31/14 主分类号 A61K38/12
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