发明名称 9-(ARYL OR HETEROARYL)-2-(PYRAZOLYL, PYRROLIDINYL OR CYCLOPENTYL)AMINOPURINE DERIVATIVES AS ANTICANCER AGENTS
摘要 Compounds of the Formula (I) in which X, R1 and R2 have the meanings indicated in Claim 1, are inhibitors of GCN2, and can be employed, inter alia, for the treatment of cancer.
申请公布号 WO2014135245(A1) 申请公布日期 2014.09.12
申请号 WO2014EP00371 申请日期 2014.02.11
申请人 MERCK PATENT GMBH 发明人 HOELZEMANN, GUENTER;DORSCH, DIETER;WEGENER, ANSGAR;POESCHKE, OLIVER;BUSCH, MICHAEL;SEENISAMY, JEYAPRAKASHNARAYANAN
分类号 C07D473/32;A61K31/52;A61P35/00 主分类号 C07D473/32
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