发明名称 |
9-(ARYL OR HETEROARYL)-2-(PYRAZOLYL, PYRROLIDINYL OR CYCLOPENTYL)AMINOPURINE DERIVATIVES AS ANTICANCER AGENTS |
摘要 |
Compounds of the Formula (I) in which X, R1 and R2 have the meanings indicated in Claim 1, are inhibitors of GCN2, and can be employed, inter alia, for the treatment of cancer. |
申请公布号 |
WO2014135245(A1) |
申请公布日期 |
2014.09.12 |
申请号 |
WO2014EP00371 |
申请日期 |
2014.02.11 |
申请人 |
MERCK PATENT GMBH |
发明人 |
HOELZEMANN, GUENTER;DORSCH, DIETER;WEGENER, ANSGAR;POESCHKE, OLIVER;BUSCH, MICHAEL;SEENISAMY, JEYAPRAKASHNARAYANAN |
分类号 |
C07D473/32;A61K31/52;A61P35/00 |
主分类号 |
C07D473/32 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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