发明名称 METHYL(R)-7-[3-AMINO-4-(2,4,5-TRIFLUOROPHENYL)-BUTYRYL]-3-TRIFLUOROMETHYL-5,6,7,8-TETRAHYDRO-IMIDAZO[1,5-a]PYRAZINE-1-CARBOXYLATE SALTS
摘要 FIELD: medicine, pharmaceutics.SUBSTANCE: invention refers to pharmaceutically acceptable (R)-7-[3-amino-4-(2,4,5-trifluorophenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1-carboxylic acid methyl ester salts specified in a group consisting of phosphate salt, hydrochloride salt, sulphate salt, mesylate salt, maleate salt or malate salt. Also, the invention refers to a method for preparing the above salts, using them and a pharmaceutical composition on the basis of the above salts.EFFECT: there are prepared new pharmaceutically acceptable (R)-7-[3-amino-4-(2,4,5-trifluorophenyl)-butyryl]-3-trifluoromethyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1-carboxylic acid methyl ester salts effective in treating diabetes.5 cl, 3 tbl, 8 ex
申请公布号 RU2528233(C2) 申请公布日期 2014.09.10
申请号 RU20110149160 申请日期 2010.04.29
申请人 TSZJANSU KHEHNZHUJ MEDITSIN KO., LTD. 发明人 JUAN' KAJKHUN;MA SHUTSIN';CHZHU LIN';LJU KHUAVEHN'
分类号 C07D471/04;A61K31/4985;A61P3/10 主分类号 C07D471/04
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