发明名称 SALT FORMS OF 4-(4-METHYLPIPERAZIN-1-YLMETHYL)-n-[4-METHYL-3-(4-PYRIDIN-3-YL)PYRIMIDIN-2-YLAMINO)PHENYL]-BENZAMIDE
摘要 <p>The present invention relates to acid addition salts of 4-[4-methyl-1-piperazinylmethyl]-N-[4-methyl-3-[[4-3-pyridinyl-2-pyrimidinyl]amino]phenyl]-benzamide, which are selected from the group consisting of a tartrate salt, such as a (D)(-) tartrate salt or a (L)(+) tartrate salt, a hydrochloride salt, a citrate sat, a malate salt, a fumarate salt, a succinate salt, a benzoate salt, a benzenesulfonate salt, a pamoate salt, a formate salt, a malonate salt, a 1,5-naphthalenedisulfonate salt, a salicylate salt, a cyclohexanesulfamate salt, a lactate salt, a mandelate salt, aq glutarate salt, an adipate salt, a squarate salt, a vanillate salt, an oxaloacetate salt, an ascorbate salt and a sulfate salt.</p>
申请公布号 PH12013500157(A1) 申请公布日期 2014.09.08
申请号 PH12013500157 申请日期 2013.01.22
申请人 NOVARTIS AG 发明人 HANS MICHAEL BURGER;PAUL WILLIAM MANLEY;MICHAEL MUTZ
分类号 A61K31/506;A61P35/00;A61P35/02;C07D401/04 主分类号 A61K31/506
代理机构 代理人
主权项
地址