发明名称 PIPERIDINYL ALKYNE OREXIN RECEPTOR ANTAGONISTS
摘要 The present invention is directed to piperidinyl alkyne compounds which are antagonists of orexin receptors. The present invention is also directed to uses of the piperidinyl alkyne compounds described herein in the treatment or prevention of neurological and psychiatric disorders and diseases in which orexin receptors are involved. The present invention is also directed to pharmaceutical compositions comprising these compounds. The present invention is also directed to uses of these pharmaceutical compositions in the prevention or treatment of such diseases in which orexin receptors are involved.
申请公布号 EP2771001(A1) 申请公布日期 2014.09.03
申请号 EP20120844517 申请日期 2012.10.19
申请人 MERCK SHARP & DOHME CORP. 发明人 KUDUK, SCOTT, D.;SKUDLAREK, JASON, W.
分类号 A61K31/4545;A61K31/4523;A61K31/454;A61K31/4709;A61P25/00;C07D401/10;C07D401/12;C07D401/14;C07D417/06;C07D417/14 主分类号 A61K31/4545
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