发明名称 |
KONDENSEREDE HETEROCYKLISKE PHENYLAMIDOFORBINDELSER TIL FOREBYGGELSE OG BEHANDLING AF GLUCOKINASE-MEDIEREDE SYGDOMME |
摘要 |
The present invention relates to a compound of formula (VIa):
or a pharmaceutically acceptable s alt or solvate thereof, wherein Ring A is pyrazinyl and L 1 , R 1 , R 1a , R 4 , L 2 , R 2 , R 3 , w and n are as defined herein. Such compounds are glucokinase agonists and useful in the treatment of diseases including diabetes and obesity. |
申请公布号 |
DK2463283(T3) |
申请公布日期 |
2014.08.18 |
申请号 |
DK20120158318T |
申请日期 |
2007.04.11 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
BAI, HAO;NUKUI, SEIJI;ZHOU, RU;BAILEY, SIMON;BHUMRALKAR, DILIP, RAMAKANT;BI, FENG;GUO, FENGLI;HE, MINGYING;HUMPHRIES, PAUL, STUART;LING, ANTHONY, LAI;LOU, JIHONG |
分类号 |
C07D401/12;A61K31/41;A61K31/435;A61K31/495;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D413/14;C07D417/12;C07D417/14 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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