发明名称 HETEROAROMATISKE OG AROMATISKE PIPERAZINYLAZETIDINYLAMIDER SOM MONOACYLGLYCEROLLIPASEINHIBITOR
摘要 Disclosed are compounds, compositions and methods for treating diseases, syndromes, conditions and disorders that are affected by the inhibition of MGL, including pain. Such compounds are represented by Formula (I) as follows: wherein Y, r, R2 and Z are defined herein.
申请公布号 DK2421852(T3) 申请公布日期 2014.08.18
申请号 DK20100719479T 申请日期 2010.04.22
申请人 JANSSEN PHARMACEUTICA N.V. 发明人 CHEVALIER, KRISTEN, M.;DAX, SCOTT, L.;FLORES, CHRISTOPHER, M.;LIU, LI;MACIELAG, MARK, J.;MCDONNELL, MARK, E.;NELEN, MARINA, I.;TODD, MATTHEW;ZHANG, SUI-PO;ZHU, BIN;NULTON, ERICA, L.;CLEMENTE, JOSE;PROUTY, STEPHEN
分类号 C07D401/12;A61K31/496;A61P25/00;A61P29/00;C07D401/14;C07D403/12;C07D403/14;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/12 主分类号 C07D401/12
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