The present invention relates to novel salt forms with improved manufacturability and solid-state properties of [6-Fluoro-1-(4-morpholin-4-ylmethyl-phenyl)-5,5-dioxo-4,5- dihydro-1 H-5l6-thiochromeno[4,3-c]pyrazol-3-yl]-morpholin-4-yl-methanone, and to methods of their manufacture.
申请公布号
WO2014121901(A1)
申请公布日期
2014.08.14
申请号
WO2014EP00205
申请日期
2014.01.27
申请人
MERCK PATENT GMBH
发明人
BECKER, AXEL;KUEHN, CLEMENS;SAAL, CHRISTOPH;DONINI, CRISTINA;VOISIN, FLORENT;MUZURELLE, MATHILDE;GERBER, PATRICK;MEDERSKI, WERNER W. K. R.;LEONARDI, ANDREA;MARIN, DELPHINE;HARRIS, LUKE