发明名称 Method of preparing (+)-1,4-dihydro-7-[(3<i>S</i>,4<i>S</i>)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid
摘要 Methods of preparing (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid are disclosed. Also provided are pharmaceutical compositions comprising (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid, and methods of treatment using such compositions.
申请公布号 US8802719(B2) 申请公布日期 2014.08.12
申请号 US201313940157 申请日期 2013.07.11
申请人 Sunesis Pharmaceuticals, Inc. 发明人 Sudhakar Anantha;Subramani Tamilarasan;Rahuman Mohamed Shiek Mohamed Mujeebur;Subbiah Ramar
分类号 A61K31/4015;C07D207/12;C07D207/14 主分类号 A61K31/4015
代理机构 Jones Day 代理人 Jones Day
主权项 1. A compound selected from
地址 South San Francisco CA US