发明名称 |
Method of preparing (+)-1,4-dihydro-7-[(3<i>S</i>,4<i>S</i>)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid |
摘要 |
Methods of preparing (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid are disclosed. Also provided are pharmaceutical compositions comprising (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid, and methods of treatment using such compositions. |
申请公布号 |
US8802719(B2) |
申请公布日期 |
2014.08.12 |
申请号 |
US201313940157 |
申请日期 |
2013.07.11 |
申请人 |
Sunesis Pharmaceuticals, Inc. |
发明人 |
Sudhakar Anantha;Subramani Tamilarasan;Rahuman Mohamed Shiek Mohamed Mujeebur;Subbiah Ramar |
分类号 |
A61K31/4015;C07D207/12;C07D207/14 |
主分类号 |
A61K31/4015 |
代理机构 |
Jones Day |
代理人 |
Jones Day |
主权项 |
1. A compound selected from |
地址 |
South San Francisco CA US |