发明名称 |
Solid Forms of 3-(6-(1-(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)Cyclopropanecarboxamido)-3-Methylpyridin-2-yl)Benzoic Acid |
摘要 |
The present invention relates to a substantially a solid form of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid (Compound 1, Solvate Form A and Compound 1, HCl Salt Form A), processes for making such forms, pharmaceutical compositions thereof, and methods of treatment therewith. |
申请公布号 |
US2014221430(A1) |
申请公布日期 |
2014.08.07 |
申请号 |
US201414250009 |
申请日期 |
2014.04.10 |
申请人 |
Vertex Pharmaceuticals Incorporated |
发明人 |
KESHAVARZ-SHOKRI Ali;ZHANG Beili;KRAWIEC Mariusz |
分类号 |
C07D405/12;A61K31/443 |
主分类号 |
C07D405/12 |
代理机构 |
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代理人 |
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主权项 |
1. A solid form of 3-(6-(1-(2,2-Difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid (Compound 1), characterized as Compound 1, Solvate Form A or Compound 1, HCl Salt Form A. |
地址 |
Boston MA US |