发明名称 Solid Forms of 3-(6-(1-(2,2-Difluorobenzo[D][1,3]Dioxol-5-yl)Cyclopropanecarboxamido)-3-Methylpyridin-2-yl)Benzoic Acid
摘要 The present invention relates to a substantially a solid form of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid (Compound 1, Solvate Form A and Compound 1, HCl Salt Form A), processes for making such forms, pharmaceutical compositions thereof, and methods of treatment therewith.
申请公布号 US2014221430(A1) 申请公布日期 2014.08.07
申请号 US201414250009 申请日期 2014.04.10
申请人 Vertex Pharmaceuticals Incorporated 发明人 KESHAVARZ-SHOKRI Ali;ZHANG Beili;KRAWIEC Mariusz
分类号 C07D405/12;A61K31/443 主分类号 C07D405/12
代理机构 代理人
主权项 1. A solid form of 3-(6-(1-(2,2-Difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid (Compound 1), characterized as Compound 1, Solvate Form A or Compound 1, HCl Salt Form A.
地址 Boston MA US