发明名称 SALT OF FUSED HETEROCYCLIC DERIVATIVE AND CRYSTAL THEREOF
摘要 An objective of the present invention is to improve the solubility of 3-[2-fluoro-5-(2,3-difluoro-6-methoxybenzyloxy)-4-methoxyphenyl]-2,4-dioxo-1,2,3,4-tetrahydrothieno[3,4-d]pyrimidine-5-carboxylic acid. The present invention provides 3-[2-fluoro-5-(2,3-difluoro-6-methoxybenzyl-oxy)-4-methoxyphenyl]-2,4-dioxo-1,2,3,4-tetrahydrothieno[3,4-d]pyrimidine-5-carboxy lic acid choline salt has excellent solubility and storage stability.
申请公布号 EP2535342(B1) 申请公布日期 2014.08.06
申请号 EP20110742250 申请日期 2011.02.09
申请人 KISSEI PHARMACEUTICAL CO., LTD. 发明人 JO, KAZUMICHI;TAKEUCHI, HIDEKI
分类号 C07D495/04;A61K31/519;A61P5/04;A61P15/08;A61P15/16;A61P15/18;A61P35/00 主分类号 C07D495/04
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