发明名称 PROCESSES FOR THE PREPARATION OF CABAZITAXEL INVOLVING C(7) -OH AND C(13) -OH SILYLATION OR JUST C(7) -OH SILYLATION
摘要 <p>The present invention discloses a process for the preparation of 4-acetoxy-2α-benzoyloxy-5β,20-epoxy-1-hydroxy-7β,10β-dimethoxy-9-oxotax-11-en-13α-yl(2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenyl-propionate Cabazitaxel (I).</p>
申请公布号 EP2760848(A1) 申请公布日期 2014.08.06
申请号 EP20120783667 申请日期 2012.09.21
申请人 FRESENIUS KABI ONCOLOGY LIMITED;LAHIRI, SASWATA;GUPTA, NITIN;AZIM, ABUL;PANDA, NILENDU;MISHRA, BHUWAN BHASKAR;SANGHANI, SUNIL 发明人 LAHIRI, SASWATA;GUPTA, NITIN;AZIM, ABUL;PANDA, NILENDU;MISHRA, BHUWAN BHASKAR;SANGHANI, SUNIL
分类号 C07D305/14;A61K31/335 主分类号 C07D305/14
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