发明名称 |
Process and intermediates for preparing integrase inhibitors |
摘要 |
The invention provides synthetic processes and synthetic intermediates that can be used to prepare 4-oxoquinolone compounds having useful integrase inhibiting properties. |
申请公布号 |
US8796459(B2) |
申请公布日期 |
2014.08.05 |
申请号 |
US201213619297 |
申请日期 |
2012.09.14 |
申请人 |
Gilead Sciences, Inc. |
发明人 |
Dowdy Eric;Chen Xi;Pfeiffer Steven |
分类号 |
A61K31/47;A61K31/4174;A61K31/216;C07D215/20;C07D233/22;C07C69/773 |
主分类号 |
A61K31/47 |
代理机构 |
Morrison & Foerster LLP |
代理人 |
Morrison & Foerster LLP ;Boss Brandon;Silver Joel |
主权项 |
1. A method of preparing a compound of formula 4: or a salt thereof comprising converting a corresponding compound of formula 3:or a salt thereof to the compound of formula 4 or the salt thereof. |
地址 |
Foster City CA US |