发明名称 Process and intermediates for preparing integrase inhibitors
摘要 The invention provides synthetic processes and synthetic intermediates that can be used to prepare 4-oxoquinolone compounds having useful integrase inhibiting properties.
申请公布号 US8796459(B2) 申请公布日期 2014.08.05
申请号 US201213619297 申请日期 2012.09.14
申请人 Gilead Sciences, Inc. 发明人 Dowdy Eric;Chen Xi;Pfeiffer Steven
分类号 A61K31/47;A61K31/4174;A61K31/216;C07D215/20;C07D233/22;C07C69/773 主分类号 A61K31/47
代理机构 Morrison & Foerster LLP 代理人 Morrison & Foerster LLP ;Boss Brandon;Silver Joel
主权项 1. A method of preparing a compound of formula 4: or a salt thereof comprising converting a corresponding compound of formula 3:or a salt thereof to the compound of formula 4 or the salt thereof.
地址 Foster City CA US