Cyclothiocarbamate derivatives as progesterone receptor modulators

摘要

Methods of using compounds which are progesterone receptor agonists for contraception and the treatment of progesterone-related maladies alone or in combination with an estrogen receptor agonist or progesterone receptor antagonist are provided. These compounds have the structure:;
wherein R1, R2, R3, R4, R5, and Q1 are defined herein.

主权项

1. A method of treating endometriosis, said method comprising delivering 5-(4,4-Dimethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile or a pharmaceutically acceptable salt thereof to a female patient.