| 发明名称 |
HAPTENS OF PALIPERIDONE |
| 摘要 |
The invention relates to compounds of Formula I, wherein L1, L2, and L3 are defined in the specification, useful for the synthesis of novel conjugates and immunogens derived from paliperidone. The invention also relates to conjugates of a paliperidone hapten and a protein.; |
| 申请公布号 |
US2014213767(A1) |
申请公布日期 |
2014.07.31 |
| 申请号 |
US201313970660 |
申请日期 |
2013.08.20 |
| 申请人 |
Ortho-Clinical Diagnostics, Inc. ;Janssen Pharmaceutica NV |
发明人 |
HASPESLAGH Pieter Rik;Vliegen Maarten;Hryhorenko Eric;DeCory Thomas R.;Sankaran Banumathi |
| 分类号 |
C07D471/04;C07K14/77;A61K47/48;C07K14/47 |
主分类号 |
C07D471/04 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
1. The compounds of Formula Iwherein
L1 is OC(O)(CH2)n, or O(CH2)n; wherein n is 1, 2, or 3; L2 is NHC(O),or absent;
L3 is (CH2)mCO2H, orwherein m is 1, 2, or 3; provided that m may only be 0 if L2 is absent. |
| 地址 |
Raritan NJ US |
