发明名称 NEW SALT AND MEDICAL USE.
摘要 The invention provides 4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2- fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide or a pharmaceutically acceptable salt thereof for the treatment of a disease associated with elevated blood uric acid levels, such as hyperuricemia or gout. In another aspect the invention provides the tosylate salt of 4-[2-(5-amino-1H-pyrazol-4- yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benz enesulfonamide.
申请公布号 MX2014004737(A) 申请公布日期 2014.07.28
申请号 MX20140004737 申请日期 2012.10.19
申请人 PFIZER LIMITED 发明人 ZAHID ALI;KENNETH JOHN BUTCHER;RICHARD PHILIP BUTT;STEPHEN JOHN FELSTEAD;SOPHIE GLATT;RUTH MITCHELL MCKERNAN;MANINDER PANESAR
分类号 A61K31/427;A61P19/06;C07D417/12 主分类号 A61K31/427
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