发明名称 Process Using Grignard Reagents
摘要 The present invention relates to a process using Grignard reagents for providing thio-triazolo group-containing compounds.
申请公布号 US2014206884(A1) 申请公布日期 2014.07.24
申请号 US201414223103 申请日期 2014.03.24
申请人 DOCHNAHL Maximilian;KEIL Michael;GEBHARDT Joachim;VOGELBACHER Uwe Josef;MENGES Frederik;RACK Michael;RENNER Jens;WOLF Bernd 发明人 DOCHNAHL Maximilian;KEIL Michael;GEBHARDT Joachim;VOGELBACHER Uwe Josef;MENGES Frederik;RACK Michael;RENNER Jens;WOLF Bernd
分类号 A01N43/653;A01N55/00 主分类号 A01N43/653
代理机构 代理人
主权项 1. A process for preparing a compound (IIIa) comprising (i) reacting a compound of formula (IV) with a Grignard reagent R1MgQ (V), wherein: R is an organic group; Q is R1 or X, wherein X is halogen; and R1 is (C1-C10)-alkyl, (C2-C10)-alkenyl, (C2-C10)-alkynyl, (C3-C8)-cycloalkyl or (C6-C10)-aryl, wherein the aryl is unsubstituted or substituted by one, two or three groups independently selected from the group consisting of halogen and (C1-C4)-alkyl.
地址 Mannheim DE