发明名称 PHARMACEUTICAL PREPARATION FOR ORAL ADMINISTRATION COMPRISING AN IMIDE COMPOUND
摘要 The present invention is directed to a preparation for oral administration comprising: a pregelatinized starch comprising N-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]-(2R,3R)-2,3-tetramethylene-butyl]-(1'R,2'S,3'R,4'S)-2,3-bicyclo[2,2,1]heptanedicarboxyimide hydrochloride (lurasidone) represented by the formula (1) as an active ingredient; a water-soluble excipient; and a water-soluble polymeric binder. The preparation exhibiting an invariant level of elution behavior even when the content of its active ingredient is varied.
申请公布号 CA2606510(C) 申请公布日期 2014.07.22
申请号 CA20062606510 申请日期 2006.05.26
申请人 DAINIPPON SUMITOMO PHARMA CO., LTD. 发明人 FUJIHARA, KAZUYUKI
分类号 A61K31/496;A61K9/20;A61K47/10;A61K47/26;A61K47/38;C07D417/12 主分类号 A61K31/496
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