发明名称 |
Process for preparing 5-fluoro-1H-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof |
摘要 |
The present invention relates to a process for the synthesis of 5-fluoro-1H-pyrazolo [3, 4-b]pyridin-3-amine in high yield and purity. The present invention also relates to processes for the synthesis of 5-fluoro-1H-pyrazolo [3, 4- b]ρyridin-3-amine derivatives. These processes are useful for preparing biologically active compounds, particularly certain GSK-3 inhibitors, or derivatives thereof. Reagents and conditi ons : i. Pd ( OAc ) |
申请公布号 |
AU2008282156(B2) |
申请公布日期 |
2014.07.17 |
申请号 |
AU20080282156 |
申请日期 |
2008.07.31 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
JIMENEZ, JUAN-MIGUEL;GAO, HUAI;HAMON, SYLVAIN LOIC JEAN-LUC;MILLER, ANDREW;DROS, ALBERT CORNELIS;COLLIER, PHILIP;GREEN, JEREMY |
分类号 |
C07D471/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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