发明名称 |
SUBSTITUTED SPIROPYRIDO[1,2-a]PYRAZINE DERIVATIVE AND MEDICINAL USE THEREOF AS HIV INTEGRASE INHIBITOR |
摘要 |
Provided is a substituted spiropyrido[1,2-a]pyrazine derivative or a pharmaceutically acceptable salt thereof which are useful as an anti-HIV agent. The invention relates to a compound represented by general formula [I] or [II] or a pharmaceutically acceptable salt thereof [in the formulae, the symbols have the same meanings as in the description]. |
申请公布号 |
WO2014104279(A1) |
申请公布日期 |
2014.07.03 |
申请号 |
WO2013JP85059 |
申请日期 |
2013.12.27 |
申请人 |
JAPAN TOBACCO INC. |
发明人 |
MIYAZAKI, SUSUMU;ISOSHIMA, HIROTAKA;OSHITA, KENGO;KAWASHITA, SEIJI;NAGAHASHI, NOBORU;TERASHITA, MASAKAZU |
分类号 |
C07D471/10;A61K31/499;A61K45/00;A61P31/18;A61P43/00;C12N15/09 |
主分类号 |
C07D471/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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