发明名称 Process for preparation of enantiomerically pure S-(+)-N, N-dimethyl-a-[2-(naphthalenyloxy)ethyl] benzenemethanamine
摘要 The present invention relates to improved, efficient process for the preparation of enantiomerically pure S-(+)-N,N-dimethyl-a-[2-(naphthalenyloxy)ethyl] benzenemethanamine and pharmaceutically acid addition salts thereof. The present invention particularly provides a process for preparation of (3S, 4R)-3-hydroxy-1-(4-methoxyphenyl)-4-phenylazetidin-2-one useful as a key intermediate for preparation of (s)-dapoxetine.
申请公布号 EP2749553(A1) 申请公布日期 2014.07.02
申请号 EP20120199791 申请日期 2012.12.31
申请人 DEVA HOLDING ANONIM SIRKETI 发明人 KOC, FIKRET;KARLIGA, BEKIR;BELLUR ATICI, ESEN;ILHAN, SUNA AYSE
分类号 C07D205/08;C07C213/06;C07C217/54 主分类号 C07D205/08
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