发明名称 PROCESS FOR THE PREPARATION OF (5-FLUORO-2-METHYL-3-QUINOLIN-2-YLMETHYL-INDOL-1-YL)-ACETIC ACID ESTERS
摘要 <p>The invention relates to a process for the preparation of a compound of formula (I) wherein R1 is C1C6 alkyl or benzyl by reacting a compound of formula (II) wherein R1 is as defined for formula (I) with 2-quinoline carboxaldehyde. The process is suitable for use on an industrial scale.</p>
申请公布号 SG11201402798R(A) 申请公布日期 2014.06.27
申请号 SG11201402798R 申请日期 2012.12.14
申请人 ATOPIX THERAPEUTICS LIMITED 发明人 TONNEL, JACQUES;PINTUS, TONY;BURGOS, ALAIN
分类号 C07D401/06 主分类号 C07D401/06
代理机构 代理人
主权项
地址