发明名称 2-OXO-OXAZOLIDIN-3,5-DIYL ANTIBIOTIC DERIVATIVES.
摘要 <p>The invention relates to antibacterial compounds of formula I (Fornula I) (I) wherein R1a represents H or carboxy and R1b represents H, or R1a and R1b represent together either the group *-C(0)-NH-S-# or the group *-C(OH)=N-S-# wherein "*" represents the point of attachment of R1a and "#" represents the point of attachment of R1b; R2 represents H, (C1-C3)alkyl, hydroxy-(C1C3)alkyl, benzyl or (C3-C5)cycloalkyl; R3 represents H or halogen; U represents N or CR4; wherein R4 is H or (C1-C3)alkoxy; A represents CH, B represents NH and m represents 1 or 2 and n represents 1 or 2; or A represents N, B is absent, m represents 2 and n represents 2; Y represents CH or N; and Q represents O or S; and salts of such compounds.</p>
申请公布号 MX2014005637(A) 申请公布日期 2014.06.23
申请号 MX20140005637 申请日期 2012.11.07
申请人 ACTELION PHARMACEUTICALS LTD 发明人 CHRISTIAN HUBSCHWERLEN;GEORG RUEEDI;CORNELIA ZUMBRUNN ACKLIN;JEAN-PHILIPPE SURIVET
分类号 C07D413/14;A61K31/501 主分类号 C07D413/14
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