发明名称 CRYSTALLINE POLYMORPHIC FORMS OF AN ANTIDIABETIC COMPOUND
摘要 The present invention relates to polymorphic forms of a compound of formula A:;;This compound is useful as a glucagon receptor antagonist and serves as a pharmaceutically active ingredient for the treatment of type 2 diabetes and related conditions, such as hyperglycemia, obesity, dyslipidemia, and the metabolic syndrome. Hydrates, hemihydrates, anhydrates and similar polymorphic forms are included.
申请公布号 US2014171480(A1) 申请公布日期 2014.06.19
申请号 US201414186829 申请日期 2014.02.21
申请人 Merck Sharp & Dohme Corp. 发明人 Chung John Y. L.;Zhang Yanfeng;Artino Laura;Cote Aaron S.;Desmond Donal;Scott Jeremy;Vaynshteyn Yekaterina
分类号 C07D209/18 主分类号 C07D209/18
代理机构 代理人
主权项 1. A crystalline polymorphic form of a compound of formula A: or a pharmaceutically acceptable salt thereof, the polymorphic form being an anhydrous free acid of polymorphic Form II.
地址 Rahway NJ US