发明名称 Selective androgen receptor modulators (SARMs) and uses thereof
摘要 Provided herein are compounds, such as compounds of Formula I, that bind to androgen receptors and/or modulate activity of androgen receptors. Also provided are methods for making and using such compounds. Also provided are compositions including such compounds and methods for making and using such compositions.;
申请公布号 US8748633(B2) 申请公布日期 2014.06.10
申请号 US201213694063 申请日期 2012.10.23
申请人 Ligand Pharmaceuticals Incorporated 发明人 Zhi Lin
分类号 C07D207/08 主分类号 C07D207/08
代理机构 代理人
主权项 1. A method for modulating an androgen receptor, comprising: contacting an androgen receptor with a compound of formula I: wherein: R1 is CF3, F or Cl;R2 is H or methyl; andR3 is H or methyl,or a pharmaceutically acceptable salt or ester thereof.
地址 La Jolla CA US