发明名称 |
PROCESS FOR THE PREPARATION OF [(1R),2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-f][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER |
摘要 |
The invention relates to an improved process for preparing [(1R),2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester of the formula (I). Compound (I) has been shown to be useful for the treatment of certain types of cancer. |
申请公布号 |
EA019693(B1) |
申请公布日期 |
2014.05.30 |
申请号 |
EA20080002171 |
申请日期 |
2007.04.19 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
CRISPINO GERARD, A.;HAMEDI MOURAD;LAPORTE THOMAS, L.;THORNTON JOHN, E.;PESTI JAAN, A.;XU ZHONGMIN;LOBBEN PAUL, C.;LEAHY DAVID, K.;MUSLEHIDDINOGLU JALE;LAI CHIAJEN;SPANGLER LORI, ANN;DISCORDIA ROBERT, P. |
分类号 |
C07D487/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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