发明名称 PROCESS FOR THE PREPARATION OF [(1R),2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-f][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
摘要 The invention relates to an improved process for preparing [(1R),2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester of the formula (I). Compound (I) has been shown to be useful for the treatment of certain types of cancer.
申请公布号 EA019693(B1) 申请公布日期 2014.05.30
申请号 EA20080002171 申请日期 2007.04.19
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 CRISPINO GERARD, A.;HAMEDI MOURAD;LAPORTE THOMAS, L.;THORNTON JOHN, E.;PESTI JAAN, A.;XU ZHONGMIN;LOBBEN PAUL, C.;LEAHY DAVID, K.;MUSLEHIDDINOGLU JALE;LAI CHIAJEN;SPANGLER LORI, ANN;DISCORDIA ROBERT, P.
分类号 C07D487/04 主分类号 C07D487/04
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