发明名称 NEW CO-CRYSTAL COMPOUND OF RIVAROXABAN AND MALONIC ACID
摘要 The present invention relates to a novel cocrystal compound of 5-chloro-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-1,3-oxazolidin-5-yl}methyl)-2-thiophenecarboxamide (rivaroxaban) and malonic acid, to processes for its preparation, to medicaments comprising this compound and to their use for controlling diseases.
申请公布号 HK1157759(A1) 申请公布日期 2014.05.30
申请号 HK20110112006 申请日期 2011.11.07
申请人 BAYER INTELLECTUAL PROPERTY GMBH 发明人 GRUNENBERG, ALFONS;FÄHNRICH, KARSTEN;QUECKENBERG, OLAF;REUTE, CHRISTIANE;KEIL, BIRGIT;GUSHURST, KAREN, SUE;STILL, EZRA, JOHN
分类号 C07D;A61K;A61P 主分类号 C07D
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