发明名称 IMPROVED PROCESS FOR PREPARING BENZOFURAN-2-CARBOXAMIDE DERIVATIVES
摘要 Provided herein are novel, commercially viable and industrially advantageous processes for the preparation of benzofuran-2-carboxamide derivatives and their intermediates, or a pharmaceutically acceptable salt thereof, in high yield and purity. Provided particularly herein are novel, commercially viable and industrially advantageous processes for the preparation of vilazodone or a pharmaceutically acceptable salt thereof in high yield and purity. Provided also herein is an improved and commercially viable process for the preparation of 3-(4-hydroxybutyl)-1H-indole-5-carbonitrile, in high yield and purity, using novel intermediate compound 3-(4-hydroxybutyryl)-1H-indole-5-carbonitrile.
申请公布号 WO2014006637(A3) 申请公布日期 2014.05.22
申请号 WO2013IN00404 申请日期 2013.07.01
申请人 SYMED LABS LIMITED;MOHAN RAO, DODDA;JITHENDER, AADEPU 发明人 MOHAN RAO, DODDA;JITHENDER, AADEPU
分类号 C07B43/06 主分类号 C07B43/06
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