发明名称 Métodos para preparar análogos nucleotídicos antivirales
摘要 Methods for isolating 9-{(R)-2-[((S)—{[(S)-1-(isopropoxycarbonyl)ethyl]amino}phenoxyphosphinyl)methoxy]propyl}adenine (compound 16): a method for preparing, in high diastereomeric purity, intermediate compounds 13 and 15: and a method for preparing intermediate compound 12: 9-{(R)-2-[((S)—{[(S)-1-(isopropoxycarbonyl)ethyl]amino}phenoxyphosphinyl)methoxy]propyl}adenine has anti-viral properties.
申请公布号 CO6940431(A2) 申请公布日期 2014.05.09
申请号 CO20140093468 申请日期 2014.05.02
申请人 GILEAD SCIENCES, INC. 发明人 COLBY DENISE A.;ROBERTS BENJAMIN JAMES;SCOTT ROBERT WILLIAM;MARTINS ANDREW ANTHONY;WHITE NICOLE S.
分类号 C07F9/6561 主分类号 C07F9/6561
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