发明名称 PYRIDONE/HYDROXYPYRIDINE 11-BETA HYDROXYSTEROID DEHYDROGENASE TYPE I INHIBITORS
摘要 Novel compounds are provided which are 11-beta-hydroxysteroid dehydrogenase type I inhibitors. 11-beta-hydroxysteroid dehydrogenase type I inhibitors are useful in treating, preventing, or slowing the progression of diseases requiring 11-beta-hydroxysteroid dehydrogenase type I inhibitor therapy. These novel compounds have the structure: enantiomers, diastereomers, solvates, salts, tautomers or prodrugs thereof wherein, A, W, X, Y and R1 are defined herein.
申请公布号 US2014128365(A1) 申请公布日期 2014.05.08
申请号 US201213667264 申请日期 2012.11.02
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 ROBL JEFFREY A.;WU SHUNG C.;YOON DAVID S.
分类号 A61K31/472;A61K31/435;A61K31/436;A61K31/4375;A61K31/439;A61K31/444;A61K31/4725;A61K31/506;A61P3/00;A61P3/04;A61P3/06;A61P3/10;A61P9/12;A61P19/02;A61P25/00;A61P27/06;A61P29/00;C07D217/26;C07D221/04;C07D401/12;C07D417/12;C07D453/00;C07D471/04;C07D491/052 主分类号 A61K31/472
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