发明名称 |
METHODS FOR INHIBITING PLATELET AGGREGATION USING GLP-1 RECEPTOR AGONISTS |
摘要 |
<p>Methods for inhibiting platelet aggregation using glucagon-like peptide-1 receptor (GLP-1R) agonists are disclosed. GLP-1 receptors are demonstrated to be expressed in platelets and/or megakaryocytes. Activation of GLP-1 receptors by GLP-1 agonists, such as GLP-1 and exendin-4, inhibited thrombm-induced platelet aggregation.</p> |
申请公布号 |
WO2014066992(A1) |
申请公布日期 |
2014.05.08 |
申请号 |
WO2013CA00939 |
申请日期 |
2013.11.04 |
申请人 |
HUSAIN, MANSOOR;CAMERON-VENDRIG, ALISON;NI, HEYU |
发明人 |
HUSAIN, MANSOOR;CAMERON-VENDRIG, ALISON;NI, HEYU |
分类号 |
A61K38/26;A61K38/16;A61P7/02;A61P9/10 |
主分类号 |
A61K38/26 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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